Assay Detail
Binding
CHEMBL926142
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of inactivated human Nav1.3 sodium channel
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Intermediate |
Target
Sodium channel protein type 3 subunit alpha (CHEMBL5163) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Sodium channel blockers.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 5.61 | 5.61 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL250699 | — | — | 1 | 5.61 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL250699 | — | IC50 | = | 2450.0 | nM | 5.61 |