Assay Detail
Binding
CHEMBL927172
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human factor 8 binding to immobilized phospholipid by surface plasmon resonance assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Design of protein membrane interaction inhibitors by virtual ligand screening, proof of concept with the C2 domain of factor V.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.08 | 5.11 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1614804 | — | — | 1 | 5.11 |
| CHEMBL261865 | — | — | 1 | 5.05 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1614804 | — | IC50 | = | 7800.0 | nM | 5.11 |
| CHEMBL261865 | — | IC50 | = | 8900.0 | nM | 5.05 |