Assay Detail
Functional
CHEMBL927526
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antitumor activity against human multidrug-resistant CEM/C2 cells by trypan blue exclusion assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | CEM/C2 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Design, synthesis, and biological evaluation of (E)-styrylbenzylsulfones as novel anticancer agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 8.00 | 8.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL254849 | — | — | 1 | 8.00 |
| CHEMBL253178 | — | — | 1 | 8.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL254849 | — | IC50 | = | 10.0 | nM | 8.00 |
| CHEMBL253178 | — | IC50 | = | 10.0 | nM | 8.00 |