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Assay Detail

CHEMBL927686

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Binding
Binding affinity to MMP2
31
Total Activities
31
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Intermediate

Target

72 kDa type IV collagenase (CHEMBL333)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Design and identification of selective HER-2 sheddase inhibitors via P1' manipulation and unconventional P2' perturbations to induce a molecular metamorphosis.
Yao W, Zhuo J, Burns DM, Li YL, Qian DQ, Zhang C, He C, Xu M, Shi E, Li Y, Marando CA, Covington MB, Yang G, Liu X, Pan M, Fridman JS, Scherle P, Wasserman ZR, Hollis G, Vaddi K, Yeleswaram S, Newton R, Friedman S, Metcalf B.
Bioorg Med Chem Lett (2008) 18 : 159 -163
PubMed 18036818 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 31 6.93 8.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL373532 1 8.30
CHEMBL375418 1 7.89
CHEMBL251884 1 7.89
CHEMBL253920 1 7.85
CHEMBL402954 1 7.68
CHEMBL403161 1 7.62
CHEMBL251847 1 7.50
CHEMBL403185 1 7.46
CHEMBL252678 1 7.43
CHEMBL251865 1 7.41
CHEMBL252877 1 7.30
CHEMBL252079 1 7.30
CHEMBL401870 1 7.28
CHEMBL404132 1 7.20
CHEMBL446457 1 7.07
CHEMBL429669 1 6.97
CHEMBL403380 1 6.80
CHEMBL221857 1 6.71
CHEMBL253256 1 6.41
CHEMBL252278 1 6.36
CHEMBL219104 1 6.35
CHEMBL442443 1 6.33
CHEMBL252442 1 6.31
CHEMBL252246 1 6.02
CHEMBL252081 1 5.96
CHEMBL253460 1 5.86
CHEMBL404170 1 5.60
CHEMBL403022 1 5.30
CHEMBL252912 1 -
CHEMBL251848 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL373532 IC50 = 5.0 nM 8.30
CHEMBL375418 IC50 = 13.0 nM 7.89
CHEMBL251884 IC50 = 13.0 nM 7.89
CHEMBL253920 IC50 = 14.0 nM 7.85
CHEMBL402954 IC50 = 21.0 nM 7.68
CHEMBL403161 IC50 = 24.0 nM 7.62
CHEMBL251847 IC50 = 32.0 nM 7.50
CHEMBL403185 IC50 = 35.0 nM 7.46
CHEMBL252678 IC50 = 37.0 nM 7.43
CHEMBL251865 IC50 = 39.0 nM 7.41
CHEMBL252877 IC50 = 50.0 nM 7.30
CHEMBL252079 IC50 = 50.0 nM 7.30
CHEMBL401870 IC50 = 53.0 nM 7.28
CHEMBL404132 IC50 = 63.0 nM 7.20
CHEMBL446457 IC50 = 86.0 nM 7.07
CHEMBL429669 IC50 = 106.0 nM 6.97
CHEMBL403380 IC50 = 159.0 nM 6.80
CHEMBL221857 IC50 = 195.0 nM 6.71
CHEMBL253256 IC50 = 391.0 nM 6.41
CHEMBL252278 IC50 = 433.0 nM 6.36
CHEMBL219104 IC50 = 446.0 nM 6.35
CHEMBL442443 IC50 = 472.0 nM 6.33
CHEMBL252442 IC50 = 488.0 nM 6.31
CHEMBL252246 IC50 = 960.0 nM 6.02
CHEMBL252081 IC50 = 1100.0 nM 5.96
CHEMBL253460 IC50 = 1387.0 nM 5.86
CHEMBL404170 IC50 = 2500.0 nM 5.60
CHEMBL403022 IC50 = 4999.0 nM 5.30
CHEMBL252912 IC50 < 5.0 nM -
CHEMBL251848 IC50 > 5000.0 nM -
CHEMBL404093 IC50 > 5000.0 nM -