Assay Detail
Functional
CHEMBL928088
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of PMA/ionomycin-induced PDG2 synthesis in human LAD2 cells
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | LAD2 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Novel prostaglandin D synthase inhibitors generated by fragment-based drug design.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1 | 5.77 | 5.77 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL261777 | — | — | 1 | 5.77 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL261777 | — | EC50 | = | 1700.0 | nM | 5.77 |