Assay Detail
Binding
CHEMBL929266
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Inhibition of bovine carboxypeptidase A
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Bos taurus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Development of potent and selective phosphinic peptide inhibitors of angiotensin-converting enzyme 2.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 7 | 7.71 | 9.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL408705 | — | — | 1 | 9.52 |
| CHEMBL260273 | — | — | 1 | 9.30 |
| CHEMBL261121 | — | — | 1 | 7.46 |
| CHEMBL261423 | — | — | 1 | 7.22 |
| CHEMBL408448 | — | — | 1 | 6.76 |
| CHEMBL409105 | — | — | 1 | 5.98 |
| CHEMBL408182 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL408705 | — | Ki | = | 0.3 | nM | 9.52 |
| CHEMBL260273 | — | Ki | = | 0.5 | nM | 9.30 |
| CHEMBL261121 | — | Ki | = | 35.0 | nM | 7.46 |
| CHEMBL261423 | — | Ki | = | 60.0 | nM | 7.22 |
| CHEMBL408448 | — | Ki | = | 175.0 | nM | 6.76 |
| CHEMBL409105 | — | Ki | = | 1050.0 | nM | 5.98 |
| CHEMBL408182 | — | Ki | > | 10000.0 | nM | - |