Assay Detail
Binding
CHEMBL929613
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of Plasmodium falciparum recombinant leucine aminopeptidase
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Plasmodium falciparum |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Leucine aminopeptidase (CHEMBL1293313) ↗| Type | SINGLE PROTEIN |
| Organism | Plasmodium falciparum 3D7 |
Publication
Individual stereoisomers of phosphinic dipeptide inhibitor of leucine aminopeptidase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 7.88 | 7.88 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL327844 | — | — | 1 | 7.88 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL327844 | — | Ki | = | 13.2 | nM | 7.88 |