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Assay Detail

CHEMBL929665

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Binding
Binding affinity to NTR1 in mouse brain membrane
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Mus musculus
Tissue Brain
Subcellular Membrane
Confidence 9 — Direct single protein target
Curated By Intermediate

Target

Neurotensin receptor type 1 (CHEMBL3570)
Type SINGLE PROTEIN
Organism Mus musculus

Publication

Peptide backbone modifications on the C-terminal hexapeptide of neurotensin.
Einsiedel J, Hübner H, Hervet M, Härterich S, Koschatzky S, Gmeiner P.
Bioorg Med Chem Lett (2008) 18 : 2013 -2018
PubMed 18276136 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 10.74 10.74

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL342252 1 10.74

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL342252 Ki = 0.018 nM 10.74