Assay Detail
Functional
CHEMBL930507
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Inhibition of ADP-induced platelet aggregation in human platelets
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | Platelet |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
P2Y1 receptor antagonists as novel antithrombotic agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 5 | 5.37 | 5.63 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL258406 | — | — | 1 | 5.63 |
| CHEMBL255306 | — | — | 1 | 5.42 |
| CHEMBL255307 | — | — | 1 | 5.39 |
| CHEMBL255308 | — | — | 1 | 5.21 |
| CHEMBL255095 | — | — | 1 | 5.21 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL258406 | — | IC50 | = | 2320.0 | nM | 5.63 |
| CHEMBL255306 | — | IC50 | = | 3850.0 | nM | 5.42 |
| CHEMBL255307 | — | IC50 | = | 4110.0 | nM | 5.39 |
| CHEMBL255308 | — | IC50 | = | 6110.0 | nM | 5.21 |
| CHEMBL255095 | — | IC50 | = | 6220.0 | nM | 5.21 |