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Assay Detail

CHEMBL930771

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Binding
Inhibition of human MMP13
30
Total Activities
30
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Collagenase 3 (CHEMBL280)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Quinazolinones and pyrido[3,4-d]pyrimidin-4-ones as orally active and specific matrix metalloproteinase-13 inhibitors for the treatment of osteoarthritis.
Li JJ, Nahra J, Johnson AR, Bunker A, O'Brien P, Yue WS, Ortwine DF, Man CF, Baragi V, Kilgore K, Dyer RD, Han HK.
J Med Chem (2008) 51 : 835 -841
PubMed 18251495 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 30 6.70 9.11

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL410029 1 9.11
CHEMBL429584 1 8.19
CHEMBL273054 1 8.01
CHEMBL270502 1 7.96
CHEMBL273113 1 7.75
CHEMBL272245 1 7.75
CHEMBL272007 1 7.67
CHEMBL409111 1 7.55
CHEMBL270050 1 7.52
CHEMBL271997 1 7.43
CHEMBL272008 1 7.34
CHEMBL429596 1 7.32
CHEMBL408646 1 7.24
CHEMBL271148 1 7.10
CHEMBL406919 1 6.92
CHEMBL429247 1 6.92
CHEMBL407090 1 6.91
CHEMBL272246 1 6.85
CHEMBL271535 1 6.74
CHEMBL429250 1 6.74
CHEMBL272866 1 6.61
CHEMBL406831 1 6.21
CHEMBL272261 1 5.77
CHEMBL410322 1 5.72
CHEMBL270481 1 5.52
CHEMBL270480 1 5.22
CHEMBL409223 1 5.00
CHEMBL272188 1 4.00
CHEMBL273114 1 4.00
CHEMBL271616 1 4.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL410029 IC50 = 0.78 nM 9.11
CHEMBL429584 IC50 = 6.5 nM 8.19
CHEMBL273054 IC50 = 9.8 nM 8.01
CHEMBL270502 IC50 = 11.0 nM 7.96
CHEMBL273113 IC50 = 18.0 nM 7.75
CHEMBL272245 IC50 = 18.0 nM 7.75
CHEMBL272007 IC50 = 21.2 nM 7.67
CHEMBL409111 IC50 = 28.0 nM 7.55
CHEMBL270050 IC50 = 30.5 nM 7.52
CHEMBL271997 IC50 = 37.0 nM 7.43
CHEMBL272008 IC50 = 46.0 nM 7.34
CHEMBL429596 IC50 = 48.0 nM 7.32
CHEMBL408646 IC50 = 57.0 nM 7.24
CHEMBL271148 IC50 = 79.0 nM 7.10
CHEMBL406919 IC50 = 120.0 nM 6.92
CHEMBL429247 IC50 = 120.0 nM 6.92
CHEMBL407090 IC50 = 122.0 nM 6.91
CHEMBL272246 IC50 = 140.0 nM 6.85
CHEMBL271535 IC50 = 184.0 nM 6.74
CHEMBL429250 IC50 = 184.0 nM 6.74
CHEMBL272866 IC50 = 244.0 nM 6.61
CHEMBL406831 IC50 = 610.0 nM 6.21
CHEMBL272261 IC50 = 1710.0 nM 5.77
CHEMBL410322 IC50 = 1900.0 nM 5.72
CHEMBL270481 IC50 = 3000.0 nM 5.52
CHEMBL270480 IC50 = 6000.0 nM 5.22
CHEMBL409223 IC50 = 10000.0 nM 5.00
CHEMBL272188 IC50 = 100000.0 nM 4.00
CHEMBL273114 IC50 = 100000.0 nM 4.00
CHEMBL271616 IC50 = 100000.0 nM 4.00