Assay Detail
Binding
CHEMBL931459
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]valsartan from human AT1 receptor expressed in CHO cells
6
Total Activities
6
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Beta-homo-amino acid scan of angiotensin IV.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Activity | 4 | - | - |
| Ki | 2 | 6.33 | 6.39 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL261120 | ANGIOTENSIN IV | — | 1 | 6.39 |
| CHEMBL260622 | — | — | 1 | 6.26 |
| CHEMBL408871 | — | — | 1 | - |
| CHEMBL261422 | — | — | 1 | - |
| CHEMBL259019 | — | — | 1 | - |
| CHEMBL248592 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL261120 | ANGIOTENSIN IV | Ki | = | 407.38 | nM | 6.39 |
| CHEMBL260622 | — | Ki | = | 549.54 | nM | 6.26 |
| CHEMBL408871 | — | Activity | - | — | - | |
| CHEMBL261422 | — | Activity | - | — | - | |
| CHEMBL259019 | — | Activity | - | — | - | |
| CHEMBL248592 | — | Activity | - | — | - |