Assay Detail
Functional
CHEMBL932831
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Effect on quorum sensing in Candida albicans assessed as inhibition of germ tube formation
13
Total Activities
13
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Candida albicans |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Influence of heterocyclic and oxime-containing farnesol analogs on quorum sensing and pathogenicity in Candida albicans.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 13 | 5.50 | 6.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL25308 | FARNESOL | — | 1 | 6.00 |
| CHEMBL401887 | — | — | 1 | 6.00 |
| CHEMBL256215 | — | — | 1 | 6.00 |
| CHEMBL258289 | — | — | 1 | 5.52 |
| CHEMBL270615 | — | — | 1 | 5.52 |
| CHEMBL428871 | — | — | 1 | 5.30 |
| CHEMBL255150 | — | — | 1 | 5.16 |
| CHEMBL404704 | — | — | 1 | 5.00 |
| CHEMBL403963 | — | — | 1 | 5.00 |
| CHEMBL273178 | — | — | 1 | - |
| CHEMBL255588 | — | — | 1 | - |
| CHEMBL404113 | — | — | 1 | - |
| CHEMBL255149 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL25308 | FARNESOL | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL401887 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL256215 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL258289 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL270615 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL428871 | — | IC50 | = | 5000.0 | nM | 5.30 |
| CHEMBL255150 | — | IC50 | = | 7000.0 | nM | 5.16 |
| CHEMBL404704 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL403963 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL273178 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL255588 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL404113 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL255149 | — | IC50 | >= | 100000.0 | nM | - |