Assay Detail
Binding
CHEMBL933019
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]DTG from mouse sigma-2 receptor in TRAMP cell membrane
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Cell Type | TRAMP |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PB183, a sigma receptor ligand, as a potential PET probe for the imaging of prostate adenocarcinoma.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 9.30 | 9.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL75286 | — | — | 1 | 9.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL75286 | — | Ki | = | 0.5 | nM | 9.30 |