Assay Detail
Binding
CHEMBL933892
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Inhibition of Aeromonas hydrophila beta lactamase CphA at pH 8.0
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Aeromonas hydrophila |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Competitive inhibitors of the CphA metallo-beta-lactamase from Aeromonas hydrophila.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 4.29 | 4.46 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL316034 | — | — | 1 | 4.46 |
| CHEMBL72628 | 2-PICOLINIC ACID | — | 1 | 4.12 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL316034 | — | Ki | = | 35000.0 | nM | 4.46 |
| CHEMBL72628 | 2-PICOLINIC ACID | Ki | = | 76000.0 | nM | 4.12 |