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Assay Detail

CHEMBL936932

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of GSK3
2
Total Activities
2
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
Fedorov O, Marsden B, Pogacic V, Rellos P, Müller S, Bullock AN, Schwaller J, Sundström M, Knapp S.
Proc Natl Acad Sci U S A (2007) 104 : 20523 -20528
PubMed 18077363 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 7.62 7.62
IC50 1 6.30 6.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL359482 1 7.62
CHEMBL75680 ALOISINE A 1 6.30

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL359482 Ki = 24.0 nM 7.62
CHEMBL75680 ALOISINE A IC50 = 500.0 nM 6.30