Assay Detail
Functional
CHEMBL937438
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Cytotoxicity against human K562 cells assessed as reduction in cellular ATP level after 48 hrs
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | K562 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Synthesis and anti-cancer activity of benzothiazole containing phthalimide on human carcinoma cell lines.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 4.49 | 4.82 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL261103 | CANTHARIDIMIDE | — | 1 | 4.82 |
| CHEMBL261567 | PHATHALIMIDE | — | 1 | 4.16 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL261103 | CANTHARIDIMIDE | IC50 | = | 15200.0 | nM | 4.82 |
| CHEMBL261567 | PHATHALIMIDE | IC50 | = | 69000.0 | nM | 4.16 |