Assay Detail
Binding
CHEMBL939302
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Inhibition of Bacillus anthracis sortase B
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Bacillus anthracis |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Activation of inhibitors by sortase triggers irreversible modification of the active site.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 4.66 | 4.85 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL264166 | — | — | 1 | 4.85 |
| CHEMBL407492 | — | — | 1 | 4.47 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL264166 | — | IC50 | = | 14000.0 | nM | 4.85 |
| CHEMBL407492 | — | IC50 | = | 34000.0 | nM | 4.47 |