Assay Detail
Binding
CHEMBL939343
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Inhibition of p34cdc2/cyclin B
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 8.40 | 8.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL23327 | PURVALANOLA | — | 1 | 8.40 |
| CHEMBL407391 | DIMETHYLADENINE | — | 1 | - |
| CHEMBL35820 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL23327 | PURVALANOLA | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL407391 | DIMETHYLADENINE | IC50 | = | 300000.0 | nM | - |
| CHEMBL35820 | — | IC50 | = | 300000.0 | nM | - |