Assay Detail
Binding
CHEMBL939356
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Binding affinity to ERK2
2
Total Activities
2
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 6.51 | 6.51 |
| Kd | 1 | 5.30 | 5.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL259551 | — | — | 1 | 6.51 |
| CHEMBL262615 | HIAZOLIDINEDIONE1 | — | 1 | 5.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL259551 | — | Ki | = | 310.0 | nM | 6.51 |
| CHEMBL262615 | HIAZOLIDINEDIONE1 | Kd | = | 5000.0 | nM | 5.30 |