Assay Detail
Binding
CHEMBL939379
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Binding affinity at PKA
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 4 | 5.92 | 7.32 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL104264 | — | — | 1 | 7.32 |
| CHEMBL406821 | — | — | 1 | 6.20 |
| CHEMBL143054 | — | — | 1 | 5.64 |
| CHEMBL429298 | — | — | 1 | 4.50 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL104264 | — | Ki | = | 48.0 | nM | 7.32 |
| CHEMBL406821 | — | Ki | = | 630.0 | nM | 6.20 |
| CHEMBL143054 | — | Ki | = | 2300.0 | nM | 5.64 |
| CHEMBL429298 | — | Ki | = | 32000.0 | nM | 4.50 |