Assay Detail
Binding
CHEMBL941185
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]CP-55-940 from human recombinant CB1 receptor expressed in COS cells
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | COS |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Total synthesis of photoactivatable or fluorescent anandamide probes: novel bioactive compounds with angiogenic activity.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 6.36 | 7.16 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL15848 | ANANDAMIDE | — | 1 | 7.16 |
| CHEMBL513597 | — | — | 1 | 5.55 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL15848 | ANANDAMIDE | Ki | = | 70.0 | nM | 7.16 |
| CHEMBL513597 | — | Ki | = | 2800.0 | nM | 5.55 |