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Assay Detail

CHEMBL943060

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Functional
DPPH radical scavenging activity
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Publication

Antioxidant phenylpropanoid-substituted epicatechins from Trichilia catigua.
Tang W, Hioki H, Harada K, Kubo M, Fukuyama Y.
J Nat Prod (2007) 70 : 2010 -2013
PubMed 18020420 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 7 5.27 5.64

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL399238 CINCHONAIN ID 1 5.64
CHEMBL251633 CINCHONAIN IC 1 5.60
CHEMBL251476 CINCHONAIN IB 1 5.29
CHEMBL437966 CATIGUANIN B 1 5.17
CHEMBL412194 CATIGUANIN A 1 5.15
CHEMBL401058 CINCHONAIN IA 1 5.03
CHEMBL206452 CATECHIN 1 5.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL399238 CINCHONAIN ID IC50 = 2300.0 nM 5.64
CHEMBL251633 CINCHONAIN IC IC50 = 2500.0 nM 5.60
CHEMBL251476 CINCHONAIN IB IC50 = 5100.0 nM 5.29
CHEMBL437966 CATIGUANIN B IC50 = 6700.0 nM 5.17
CHEMBL412194 CATIGUANIN A IC50 = 7100.0 nM 5.15
CHEMBL401058 CINCHONAIN IA IC50 = 9400.0 nM 5.03
CHEMBL206452 CATECHIN IC50 = 10000.0 nM 5.00