Assay Detail
Functional
CHEMBL943672
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Agonist activity at GPR40 expressed in CHO cells by FLIPR assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Cell Type | CHO |
| Confidence | 8 — Homologous single protein target |
| Curated By | Intermediate |
Publication
Discovery of diacylphloroglucinols as a new class of GPR40 (FFAR1) agonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 10.00 | 10.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL475027 | — | — | 1 | 10.00 |
| CHEMBL475054 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL475027 | — | EC50 | = | 0.1 | nM | 10.00 |
| CHEMBL475054 | — | EC50 | < | 100.0 | nM | - |