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Assay Detail

CHEMBL944126

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiproliferative activity against human NCI-H460 cells by MTT assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type NCI-H460
Confidence 1 — Organism
Curated By Autocuration

Target

NCI-H460 (CHEMBL396)
Type CELL-LINE
Organism Homo sapiens

Publication

Uncovering biosynthetic potential of plant-associated fungi: effect of culture conditions on metabolite production by Paraphaeosphaeria quadriseptata and Chaetomium chiversii.
Paranagama PA, Wijeratne EM, Gunatilaka AA.
J Nat Prod (2007) 70 : 1939 -1945
PubMed 18052326 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 6.82 8.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL53463 DOXORUBICIN 4.0 1 8.00
CHEMBL252324 1 6.52
CHEMBL215853 MONOCILLIN I 1 6.46
CHEMBL404204 MONOCILLIN III 1 6.30

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL53463 DOXORUBICIN IC50 = 10.0 nM 8.00
CHEMBL252324 IC50 = 300.0 nM 6.52
CHEMBL215853 MONOCILLIN I IC50 = 350.0 nM 6.46
CHEMBL404204 MONOCILLIN III IC50 = 500.0 nM 6.30