Assay Detail
Functional
CHEMBL944393
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Inhibition of human MDA-MB-231 cell proliferation assessed as cell viability after 48 hrs by ATPlite assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | MDA-MB-231 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Fragment-based design of small molecule X-linked inhibitor of apoptosis protein inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 4.79 | 4.79 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL458358 | — | — | 1 | 4.79 |
| CHEMBL234346 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL458358 | — | IC50 | = | 16400.0 | nM | 4.79 |
| CHEMBL234346 | — | IC50 | > | 50000.0 | nM | - |