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Assay Detail

CHEMBL946944

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Inhibition of LPS-induced TNFalpha production in human PBMC
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type PBMC
Confidence 1 — Organism
Curated By Autocuration

Target

PBMC (CHEMBL613107)
Type CELL-LINE
Organism Homo sapiens

Publication

Biphenyl amide p38 kinase inhibitors 2: Optimisation and SAR.
Angell RM, Angell TD, Bamborough P, Brown D, Brown M, Buckton JB, Cockerill SG, Edwards CD, Jones KL, Longstaff T, Smee PA, Smith KJ, Somers DO, Walker AL, Willson M.
Bioorg Med Chem Lett (2008) 18 : 324 -328
PubMed 17981461 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.60 5.60

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL273158 1 5.60

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL273158 IC50 = 2500.0 nM 5.60