Assay Detail
Binding
CHEMBL947977
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of FGFR by HTRF assay
3
Total Activities
3
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
3-amino-benzo[d]isoxazoles as novel multitargeted inhibitors of receptor tyrosine kinases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Activity | 2 | - | - |
| IC50 | 1 | 5.52 | 5.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL430090 | — | — | 1 | 5.52 |
| CHEMBL270084 | — | — | 1 | - |
| CHEMBL269884 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL430090 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL270084 | — | Activity | - | — | - | |
| CHEMBL269884 | — | Activity | - | — | - |