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Assay Detail

CHEMBL948565

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Displacement of [3H]PDBu from rat brain PKC by scintillation counting
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Rattus norvegicus
Confidence 5 — Multiple protein complex / RNA
Curated By Autocuration

Target

Protein kinase C (PKC) (CHEMBL2094266)
Type PROTEIN FAMILY
Organism Rattus norvegicus

Publication

Verbascoside isolated from Lantana camara, an inhibitor of protein kinase C.
Herbert JM, Maffrand JP, Taoubi K, Augereau JM, Fouraste I, Gleye J.
J Nat Prod (1991) 54 : 1595 -1600
PubMed 1812212 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 7.17 7.17

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL444478 ACETOSIDE 2.0 1 7.17

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL444478 ACETOSIDE IC50 = 68.0 nM 7.17