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Assay Detail

CHEMBL949121

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Functional
Antiviral activity against human rhinovirus 14
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism rhinovirus B14
Confidence 1 — Organism
Curated By Intermediate

Target

rhinovirus B14 (CHEMBL613759)
Type ORGANISM
Organism rhinovirus B14

Publication

Inhibitors of proteases and amide hydrolases that employ an alpha-ketoheterocycle as a key enabling functionality.
Maryanoff BE, Costanzo MJ.
Bioorg Med Chem (2008) 16 : 1562 -1595
PubMed 18053726 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 5 5.62 6.47

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL145753 1 6.47
CHEMBL272994 1 5.50
CHEMBL228200 1 5.40
CHEMBL402559 1 5.10
CHEMBL256829 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL145753 EC50 = 340.0 nM 6.47
CHEMBL272994 EC50 = 3200.0 nM 5.50
CHEMBL228200 EC50 = 4000.0 nM 5.40
CHEMBL402559 EC50 = 7900.0 nM 5.10
CHEMBL256829 EC50 > 10000.0 nM -