Assay Detail
Binding
CHEMBL950208
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Inhibition of CaMK2delta using 3 weeks old stock solution of compound
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Calcium/calmodulin-dependent protein kinase type II subunit delta (CHEMBL2801) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Aryl-indolyl maleimides as inhibitors of CaMKIIdelta. Part 3: Importance of the indole orientation.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.64 | 6.64 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL256827 | — | — | 1 | 6.64 |
| CHEMBL258290 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL256827 | — | IC50 | = | 230.0 | nM | 6.64 |
| CHEMBL258290 | — | IC50 | < | 39.0 | nM | - |