Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL958771

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of aromatase
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Intermediate

Target

Aromatase (CHEMBL1978)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Selective inhibition of aromatase by a dihydroisocoumarin from Xyris pterygoblephara.
Endringer DC, Guimarães KG, Kondratyuk TP, Pezzuto JM, Braga FC.
J Nat Prod (2008) 71 : 1082 -1084
PubMed 18462007 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.30 5.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL451532 NARINGIN 1 5.30

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL451532 NARINGIN IC50 = 5000.0 nM 5.30