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Assay Detail

CHEMBL959129

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Activity at human GnRH receptor by inositol phosphate functional assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Gonadotropin-releasing hormone receptor (CHEMBL1855)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Non-peptide gonadotropin-releasing hormone receptor antagonists.
Betz SF, Zhu YF, Chen C, Struthers RS.
J Med Chem (2008) 51 : 3331 -3348
PubMed 18419112 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 9.00 9.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL120432 1 9.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL120432 IC50 = 1.0 nM 9.00