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Assay Detail

CHEMBL960392

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of CDK2/Cyclin A
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

ATP competitive inhibitors of D-alanine-D-alanine ligase based on protein kinase inhibitor scaffolds.
Triola G, Wetzel S, Ellinger B, Koch MA, Hübel K, Rauh D, Waldmann H.
Bioorg Med Chem (2009) 17 : 1079 -1087
PubMed 18321716 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.16 5.16

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL280074 OLOMOUCINE 1 5.16

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL280074 OLOMOUCINE IC50 = 7000.0 nM 5.16