Assay Detail
Binding
CHEMBL963041
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Equilibrium binding affinity to wild type human PNP
10
Total Activities
10
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Immucillins in custom catalytic-site cavities.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 5 | 10.64 | 10.97 |
| Activity | 5 | - | - |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL269864 | ULODESINE | 2.0 | 1 | 10.97 |
| CHEMBL514795 | — | — | 1 | 10.71 |
| CHEMBL218291 | FORODESINE | 4.0 | 1 | 10.24 |
| CHEMBL462398 | — | — | 1 | - |
| CHEMBL505564 | — | — | 1 | - |
| CHEMBL512051 | — | — | 1 | - |
| CHEMBL461527 | — | — | 1 | - |
| CHEMBL443968 | — | — | 1 | - |
| CHEMBL474328 | — | — | 1 | - |
| CHEMBL473929 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL269864 | ULODESINE | Ki | = | 0.0107 | nM | 10.97 |
| CHEMBL514795 | — | Ki | = | 0.0196 | nM | 10.71 |
| CHEMBL218291 | FORODESINE | Ki | = | 0.0579 | nM | 10.24 |
| CHEMBL462398 | — | Activity | - | — | - | |
| CHEMBL505564 | — | Ki | = | 0.0052 | nM | - |
| CHEMBL512051 | — | Activity | - | — | - | |
| CHEMBL461527 | — | Activity | - | — | - | |
| CHEMBL443968 | — | Ki | = | 0.0098 | nM | - |
| CHEMBL474328 | — | Activity | - | — | - | |
| CHEMBL473929 | — | Activity | - | — | - |