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Assay Detail

CHEMBL963731

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of Plasmodium falciparum Pfnek1
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Plasmodium falciparum
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Alisiaquinones and alisiaquinol, dual inhibitors of Plasmodium falciparum enzyme targets from a New Caledonian deep water sponge.
Desoubzdanne D, Marcourt L, Raux R, Chevalley S, Dorin D, Doerig C, Valentin A, Ausseil F, Debitus C.
J Nat Prod (2008) 71 : 1189 -1192
PubMed 18512987 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 6.00 6.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL510492 XESTOQUINONE 1 6.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL510492 XESTOQUINONE IC50 = 1000.0 nM 6.00