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Assay Detail

CHEMBL964474

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of Cochliobolus lunatus CYP53A15 expressed in Escherichia coli
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Curvularia lunata
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

CYP53A15 of Cochliobolus lunatus, a target for natural antifungal compounds.
Podobnik B, Stojan J, Lah L, Krasevec N, Seliskar M, Rizner TL, Rozman D, Komel R.
J Med Chem (2008) 51 : 3480 -3486
PubMed 18505250 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 4 4.76 5.09

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL29411 THYMOL 2.0 1 5.09
CHEMBL445206 ISOEUGENOL 1 4.85
CHEMBL42710 EUGENOL 0.5 1 4.58
CHEMBL13883 VANILLIN -1.0 1 4.53

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL29411 THYMOL Ki = 8200.0 nM 5.09
CHEMBL445206 ISOEUGENOL Ki = 14200.0 nM 4.85
CHEMBL42710 EUGENOL Ki = 26200.0 nM 4.58
CHEMBL13883 VANILLIN Ki = 29700.0 nM 4.53