Assay Detail
Functional
CHEMBL965539
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Inhibition of CD40L, IFN-gamma and IL18 mixture-induced IL12p40 production in mouse DC-B cells after 18 to 24 hrs by fluorescence immunoassay
20
Total Activities
20
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Salicylanilides: selective inhibitors of interleukin-12p40 production.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 20 | 6.75 | 7.89 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL459303 | — | — | 1 | 7.89 |
| CHEMBL453897 | — | — | 1 | 7.89 |
| CHEMBL461545 | — | — | 1 | 7.35 |
| CHEMBL455225 | — | — | 1 | 7.13 |
| CHEMBL461542 | — | — | 1 | 6.92 |
| CHEMBL100633 | — | — | 1 | 6.89 |
| CHEMBL462415 | — | — | 1 | 6.70 |
| CHEMBL460305 | — | — | 1 | 6.62 |
| CHEMBL462592 | — | — | 1 | 6.55 |
| CHEMBL462604 | — | — | 1 | 6.50 |
| CHEMBL462603 | — | — | 1 | 6.39 |
| CHEMBL507038 | — | — | 1 | 5.57 |
| CHEMBL460481 | — | — | 1 | 5.29 |
| CHEMBL458878 | — | — | 1 | - |
| CHEMBL389507 | OSALMID | 2.0 | 1 | - |
| CHEMBL462416 | — | — | 1 | - |
| CHEMBL513453 | — | — | 1 | - |
| CHEMBL462591 | — | — | 1 | - |
| CHEMBL461733 | — | — | 1 | - |
| CHEMBL505876 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL459303 | — | IC50 | = | 13.0 | nM | 7.89 |
| CHEMBL453897 | — | IC50 | = | 13.0 | nM | 7.89 |
| CHEMBL461545 | — | IC50 | = | 45.0 | nM | 7.35 |
| CHEMBL455225 | — | IC50 | = | 74.0 | nM | 7.13 |
| CHEMBL461542 | — | IC50 | = | 120.0 | nM | 6.92 |
| CHEMBL100633 | — | IC50 | = | 130.0 | nM | 6.89 |
| CHEMBL462415 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL460305 | — | IC50 | = | 240.0 | nM | 6.62 |
| CHEMBL462592 | — | IC50 | = | 280.0 | nM | 6.55 |
| CHEMBL462604 | — | IC50 | = | 320.0 | nM | 6.50 |
| CHEMBL462603 | — | IC50 | = | 410.0 | nM | 6.39 |
| CHEMBL507038 | — | IC50 | = | 2700.0 | nM | 5.57 |
| CHEMBL460481 | — | IC50 | = | 5100.0 | nM | 5.29 |
| CHEMBL458878 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL389507 | OSALMID | IC50 | > | 10000.0 | nM | - |
| CHEMBL462416 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL513453 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL462591 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL461733 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL505876 | — | IC50 | > | 10000.0 | nM | - |