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Assay Detail

CHEMBL966027

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Phytotoxicity against Echinochloa crus-galli assessed as inhibition of radicle elongation by petri dish bioassay
19
Total Activities
15
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Echinochloa crus-galli
Confidence 1 — Organism
Curated By Autocuration

Target

Echinochloa crus-galli (CHEMBL612343)
Type ORGANISM
Organism Echinochloa crus-galli

Publication

Phytotoxic compounds from Prionosciadium watsoni.
Valencia-Islas N, Abbas H, Bye R, Toscano R, Mata R.
J Nat Prod (2002) 65 : 828 -834
PubMed 12088423 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 15 4.87 5.21
Activity 4 - -

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL463444 2 5.21
CHEMBL518222 1 4.83
CHEMBL458524 1 4.58
CHEMBL464293 1 -
CHEMBL518224 1 -
CHEMBL463449 1 -
CHEMBL70302 SERAVSHANIN 1 -
CHEMBL512733 QUIANHUCOUMARIN D 1 -
CHEMBL68727 1 -
CHEMBL457257 JATAMANSIN 1 -
CHEMBL449490 1 -
CHEMBL463635 2 -
CHEMBL503137 (+)-LOMATIN 2 -
CHEMBL464886 2 -
CHEMBL367623 2,4-DICHLOROPHENOXYACETIC ACID 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL463444 IC50 = 6190.0 nM 5.21
CHEMBL518222 IC50 = 14800.0 nM 4.83
CHEMBL458524 IC50 = 26400.0 nM 4.58
CHEMBL518224 IC50 = 595000.0 nM -
CHEMBL463449 IC50 = 155000.0 nM -
CHEMBL70302 SERAVSHANIN IC50 = 162000.0 nM -
CHEMBL512733 QUIANHUCOUMARIN D IC50 - -
CHEMBL68727 IC50 = 439000.0 nM -
CHEMBL457257 JATAMANSIN IC50 = 863000.0 nM -
CHEMBL449490 IC50 = 169000.0 nM -
CHEMBL463635 IC50 = 808000.0 nM -
CHEMBL503137 (+)-LOMATIN IC50 = 296000.0 nM -
CHEMBL464886 IC50 = 461000.0 nM -
CHEMBL367623 2,4-DICHLOROPHENOXYACETIC ACID IC50 > 220000.0 nM -
CHEMBL463444 Activity - -
CHEMBL463635 Activity - -
CHEMBL503137 (+)-LOMATIN Activity - -
CHEMBL464293 IC50 = 439000.0 nM -
CHEMBL464886 Activity - -