Assay Detail
Binding
CHEMBL969706
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Inhibition of HDAC
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Design, synthesis and biological evaluation of novel compounds with conjugated structure as anti-tumor agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.78 | 7.80 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL314389 | OXAMFLATIN | — | 1 | 7.80 |
| CHEMBL159249 | — | — | 1 | 5.75 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL314389 | OXAMFLATIN | IC50 | = | 15.7 | nM | 7.80 |
| CHEMBL159249 | — | IC50 | = | 1800.0 | nM | 5.75 |