Assay Detail
Binding
CHEMBL970659
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Inhibition of FGFRK2
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Intermediate |
Publication
Design, synthesis, and biological evaluation of potent c-Met inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 6.85 | 6.85 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL453737 | — | — | 1 | 6.85 |
| CHEMBL505896 | — | — | 1 | - |
| CHEMBL447602 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL453737 | — | IC50 | = | 140.0 | nM | 6.85 |
| CHEMBL505896 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL447602 | — | IC50 | - | — | - |