Assay Detail
Binding
CHEMBL970979
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Inhibition of CK2
7
Total Activities
5
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
A common protein fold topology shared by flavonoid biosynthetic enzymes and therapeutic targets.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 5 | 5.97 | 6.46 |
| Ki | 2 | 6.07 | 6.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL31574 | FISETIN | 2.0 | 1 | 6.46 |
| CHEMBL50 | QUERCETIN | 3.0 | 1 | 6.26 |
| CHEMBL164 | MYRICETIN | — | 2 | 6.22 |
| CHEMBL28 | APIGENIN | — | 1 | 6.10 |
| CHEMBL165 | RESVERATROL | 3.0 | 2 | 5.92 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL31574 | FISETIN | IC50 | = | 350.0 | nM | 6.46 |
| CHEMBL50 | QUERCETIN | IC50 | = | 550.0 | nM | 6.26 |
| CHEMBL164 | MYRICETIN | Ki | = | 600.0 | nM | 6.22 |
| CHEMBL28 | APIGENIN | IC50 | = | 800.0 | nM | 6.10 |
| CHEMBL164 | MYRICETIN | IC50 | = | 920.0 | nM | 6.04 |
| CHEMBL165 | RESVERATROL | Ki | = | 1200.0 | nM | 5.92 |
| CHEMBL165 | RESVERATROL | IC50 | = | 10000.0 | nM | 5.00 |