Assay Detail
Binding
CHEMBL971454
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Inhibition of baboon liver MAOB
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Papio hamadryas |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Inhibition of monoamine oxidase by (E)-styrylisatin analogues.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 5 | 6.80 | 7.68 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL447307 | — | — | 1 | 7.68 |
| CHEMBL506301 | — | — | 1 | 7.52 |
| CHEMBL466872 | — | — | 1 | 7.38 |
| CHEMBL450239 | (E)-6-STYRYLISATIN | — | 1 | 6.35 |
| CHEMBL326294 | ISATIN | — | 1 | 5.07 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL447307 | — | IC50 | = | 20.7 | nM | 7.68 |
| CHEMBL506301 | — | IC50 | = | 30.1 | nM | 7.52 |
| CHEMBL466872 | — | IC50 | = | 41.7 | nM | 7.38 |
| CHEMBL450239 | (E)-6-STYRYLISATIN | IC50 | = | 444.0 | nM | 6.35 |
| CHEMBL326294 | ISATIN | IC50 | = | 8566.0 | nM | 5.07 |