Assay Detail
Binding
CHEMBL972371
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Inhibition of human MAOB 1199A mutant
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Inhibition of monoamine oxidase by (E)-styrylisatin analogues.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 5 | 5.36 | 5.96 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL466872 | — | — | 1 | 5.96 |
| CHEMBL450239 | (E)-6-STYRYLISATIN | — | 1 | 5.66 |
| CHEMBL506301 | — | — | 1 | 5.35 |
| CHEMBL326294 | ISATIN | — | 1 | 4.92 |
| CHEMBL447307 | — | — | 1 | 4.90 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL466872 | — | Ki | = | 1100.0 | nM | 5.96 |
| CHEMBL450239 | (E)-6-STYRYLISATIN | Ki | = | 2200.0 | nM | 5.66 |
| CHEMBL506301 | — | Ki | = | 4500.0 | nM | 5.35 |
| CHEMBL326294 | ISATIN | Ki | = | 12000.0 | nM | 4.92 |
| CHEMBL447307 | — | Ki | = | 12500.0 | nM | 4.90 |