Assay Detail
Binding
CHEMBL973556
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Displacement of [3H]clonidine from Imidazoline receptor 1 rat PC-12 cells
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Cell Type | PC-12 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Novel ligands rationally designed for characterizing I2-imidazoline binding sites nature and functions.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 5.32 | 5.43 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL14210 | PHENYZOLINE | — | 1 | 5.43 |
| CHEMBL501690 | — | — | 1 | 5.20 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL14210 | PHENYZOLINE | Ki | = | 3697.0 | nM | 5.43 |
| CHEMBL501690 | — | Ki | = | 6340.0 | nM | 5.20 |