Assay Detail
Binding
CHEMBL973557
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Binding affinity to Imidazoline receptor 2
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Novel ligands rationally designed for characterizing I2-imidazoline binding sites nature and functions.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 7.70 | 8.60 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL14210 | PHENYZOLINE | — | 1 | 8.60 |
| CHEMBL501690 | — | — | 1 | 6.80 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL14210 | PHENYZOLINE | Ki | = | 2.512 | nM | 8.60 |
| CHEMBL501690 | — | Ki | = | 158.49 | nM | 6.80 |