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Assay Detail

CHEMBL980501

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiplasmodial activity against chloroquine-sensitive Plasmodium falciparum Ghana by LDH reporter assay
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Plasmodium falciparum
Confidence 1 — Organism
Curated By Autocuration

Target

Plasmodium falciparum (CHEMBL364)
Type ORGANISM
Organism Plasmodium falciparum

Publication

Antiparasitic activity of some xanthones and biflavonoids from the root bark of Garcinia livingstonei.
Mbwambo ZH, Kapingu MC, Moshi MJ, Machumi F, Apers S, Cos P, Ferreira D, Marais JP, Vanden Berghe D, Maes L, Vlietinck A, Pieters L.
J Nat Prod (2006) 69 : 369 -372
PubMed 16562837 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 7 4.70 5.22

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL500482 1 5.22
CHEMBL454538 GARCILIVIN A 1 5.17
CHEMBL188061 1 5.00
CHEMBL463023 VOLKENSIFLAVONE 1 4.32
CHEMBL479289 1 4.28
CHEMBL482023 1 4.23
CHEMBL499445 GARCIVILIN C 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL500482 IC50 = 6000.0 nM 5.22
CHEMBL454538 GARCILIVIN A IC50 = 6700.0 nM 5.17
CHEMBL188061 IC50 = 10000.0 nM 5.00
CHEMBL463023 VOLKENSIFLAVONE IC50 = 48000.0 nM 4.32
CHEMBL479289 IC50 = 52000.0 nM 4.28
CHEMBL482023 IC50 = 59000.0 nM 4.23
CHEMBL499445 GARCIVILIN C IC50 > 64000.0 nM -