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Assay Detail

CHEMBL980771

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Displacement of radioligand from dopamine D3 receptor
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Intermediate

Target

D(3) dopamine receptor (CHEMBL234)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Highly functionalized 7-azaindoles as selective PPAR gamma modulators.
Debenham SD, Chan A, Lau FW, Liu W, Wood HB, Lemme K, Colwell L, Habulihaz B, Akiyama TE, Einstein M, Doebber TW, Sharma N, Wang CF, Wu M, Berger JP, Meinke PT.
Bioorg Med Chem Lett (2008) 18 : 4798 -4801
PubMed 18701276 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 6.08 6.08

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL461571 1 6.08

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL461571 IC50 = 837.0 nM 6.08