Assay Detail
Binding
CHEMBL981116
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Inhibition of prostaglandin DP receptor
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Intermediate |
Publication
The many roles for fluorine in medicinal chemistry.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 8.93 | 9.24 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL221007 | DIASTEREOMER 2 | — | 1 | 9.24 |
| CHEMBL518461 | — | — | 1 | 8.96 |
| CHEMBL383484 | — | — | 1 | 8.59 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL221007 | DIASTEREOMER 2 | Ki | = | 0.57 | nM | 9.24 |
| CHEMBL518461 | — | Ki | = | 1.1 | nM | 8.96 |
| CHEMBL383484 | — | Ki | = | 2.6 | nM | 8.59 |