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Assay Detail

CHEMBL982908

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of HIV1 recombinant protease L10I/I15V/E35D/N37S/R41K/I62V/L63P/A71V/G73S/L90M mutant expressed in Escherichia coli by spectrophotometric assay
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Human immunodeficiency virus 1
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Human immunodeficiency virus type 1 protease (CHEMBL243)
Type SINGLE PROTEIN
Organism Human immunodeficiency virus 1

Publication

Inorganic polyhedral metallacarborane inhibitors of HIV protease: a new approach to overcoming antiviral resistance.
Kozísek M, Cígler P, Lepsík M, Fanfrlík J, Rezácová P, Brynda J, Pokorná J, Plesek J, Grüner B, Grantz Sasková K, Václavíková J, Král V, Konvalinka J.
J Med Chem (2008) 51 : 4839 -4843
PubMed 18598016 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 7 9.41 10.82

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1323 DARUNAVIR 4.0 1 10.82
CHEMBL729 LOPINAVIR 4.0 1 10.54
CHEMBL1163 ATAZANAVIR 4.0 1 10.12
CHEMBL116 AMPRENAVIR 4.0 1 9.82
CHEMBL584 NELFINAVIR 4.0 1 8.68
CHEMBL114 SAQUINAVIR 4.0 1 8.54
CHEMBL5483011 INDINAVIR 3.0 1 7.33

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1323 DARUNAVIR Ki = 0.015 nM 10.82
CHEMBL729 LOPINAVIR Ki = 0.029 nM 10.54
CHEMBL1163 ATAZANAVIR Ki = 0.076 nM 10.12
CHEMBL116 AMPRENAVIR Ki = 0.15 nM 9.82
CHEMBL584 NELFINAVIR Ki = 2.1 nM 8.68
CHEMBL114 SAQUINAVIR Ki = 2.9 nM 8.54
CHEMBL5483011 INDINAVIR Ki = 47.0 nM 7.33