Assay Detail

CHEMBL983902

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding

Inhibition of somatostatin receptor

ChEMBL ↗

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Target

Unchecked (CHEMBL612545) ↗

Open DB target context

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Unchecked (CHEMBL612545) is the working anchor for this assay review. Loading the live Open DB target snapshot…

Primary target Unchecked

CHEMBL612545

Anchored from Assay target.

Protein identity Unchecked

Disease frame Disease evidence pending

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Review focus Open DB context pending

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Total Activities

Compounds Tested

Activity Types

Assay Parameters

Assay Information

Assay Type	Binding
Confidence	0 — Uncurated / Unknown
Curated By	Autocuration

Target

Unchecked (CHEMBL612545) ↗

Type

UNCHECKED

Publication

Identification of a potent, selective, and orally active leukotriene a4 hydrolase inhibitor with anti-inflammatory activity.

Grice CA, Tays KL, Savall BM, Wei J, Butler CR, Axe FU, Bembenek SD, Fourie AM, Dunford PJ, Lundeen K, Coles F, Xue X, Riley JP, Williams KN, Karlsson L, Edwards JP.
J Med Chem (2008) 51 : 4150 -4169
PubMed 18588282 · DOI

Activity Statistics

Type	Count	Avg pChEMBL	Best pChEMBL
IC50	1	9.92	9.92

Compounds Tested

Compound	Name	Phase	Activities	Best pChEMBL
CHEMBL1823872	SOMATOSTATIN	3.0	1	9.92

Activity Data

Compound	Name	Type	Rel.	Value	Units	pChEMBL
CHEMBL1823872	SOMATOSTATIN	IC50	=	0.12	nM	9.92